Overview
| Uniprot ID | O95479 |
| Protein Name | GDH/6PGL endoplasmic bifunctional protein |
| Gene Name | H6PD |
| Organism | Homo sapiens |
Kla Sites from experimental identification
| Position |
Flanking peptide |
| 208 |
RVDHYLGKQAVAQIL |
| 293 |
AEAVLRHKLQVFQAL |
Function
Bifunctional enzyme localized in the lumen of the endoplasmic reticulum that catalyzes the first two steps of the oxidative branch of the pentose phosphate pathway/shunt, an alternative to glycolysis and a major source of reducing power and metabolic intermediates for biosynthetic processes (By similarity). Has a hexose-6-phosphate dehydrogenase activity, with broad substrate specificity compared to glucose-6-phosphate 1-dehydrogenase/G6PD, and catalyzes the first step of the pentose phosphate pathway (PubMed:12858176, PubMed:18628520, PubMed:23132696). In addition, acts as a 6-phosphogluconolactonase and catalyzes the second step of the pentose phosphate pathway (By similarity). May have a dehydrogenase activity for alternative substrates including glucosamine 6-phosphate and glucose 6-sulfate (By similarity). The main function of this enzyme is to provide reducing equivalents such as NADPH to maintain the adequate levels of reductive cofactors in the oxidizing environment of the endoplasmic reticulum (PubMed:12858176, PubMed:18628520, PubMed:23132696). By producing NADPH that is needed by reductases of the lumen of the endoplasmic reticulum like corticosteroid 11-beta-dehydrogenase isozyme 1/HSD11B1, indirectly regulates their activity (PubMed:18628520)
Protein Sequence
10
MWNMLIVAMC
20
LALLGCLQAQ
30
ELQGHVSIIL
40
LGATGDLAKK
50
YLWQGLFQLY
60
LDEAGRGHSF
70
SFHGAALTAP
80
KQGQELMAKA
90
LESLSCPKDM
100
APSHCAEHKD
110
QFLQLSQYRQ
120
LKTAEDYQAL
130
NKDIEAQLQH
140
AGLREAGRIF
150
YFSVPPFAYE
160
DIARNINSSC
170
RPGPGAWLRV
180
VLEKPFGHDH
190
FSAQQLATEL
200
GTFFQEEEMY
210
RVDHYLGKQA
220
VAQILPFRDQ
230
NRKALDGLWN
240
RHHVERVEII
250
MKETVDAEGR
260
TSFYEEYGVI
270
RDVLQNHLTE
280
VLTLVAMELP
290
HNVSSAEAVL
300
RHKLQVFQAL
310
RGLQRGSAVV
320
GQYQSYSEQV
330
RRELQKPDSF
340
HSLTPTFAAV
350
LVHIDNLRWE
360
GVPFILMSGK
370
ALDERVGYAR
380
ILFKNQACCV
390
QSEKHWAAAQ
400
SQCLPRQLVF
410
HIGHGDLGSP
420
AVLVSRNLFR
430
PSLPSSWKEM
440
EGPPGLRLFG
450
SPLSDYYAYS
460
PVRERDAHSV
470
LLSHIFHGRK
480
NFFITTENLL
490
ASWNFWTPLL
500
ESLAHKAPRL
510
YPGGAENGRL
520
LDFEFSSGRL
530
FFSQQQPEQL
540
VPGPGPAPMP
550
SDFQVLRAKY
560
RESPLVSAWS
570
EELISKLAND
580
IEATAVRAVR
590
RFGQFHLALS
600
GGSSPVALFQ
610
QLATAHYGFP
620
WAHTHLWLVD
630
ERCVPLSDPE
640
SNFQGLQAHL
650
LQHVRIPYYN
660
IHPMPVHLQQ
670
RLCAEEDQGA
680
QIYAREISAL
690
VANSSFDLVL
700
LGMGADGHTA
710
SLFPQSPTGL
720
DGEQLVVLTT
730
SPSQPHRRMS
740
LSLPLINRAK
750
KVAVLVMGRM
760
KREITTLVSR
770
VGHEPKKWPI
780
SGVLPHSGQL
790
VWYMDYDAFL
G
Gene Ontology
| Classification |
GO ID |
Description |
| Cellular Component |
GO:0005783 |
endoplasmic reticulum |
| Cellular Component |
GO:0005788 |
endoplasmic reticulum lumen |
| Cellular Component |
GO:0016529 |
sarcoplasmic reticulum |
| Molecular Function |
GO:0017057 |
6-phosphogluconolactonase activity |
| Molecular Function |
GO:0030246 |
carbohydrate binding |
| Molecular Function |
GO:0047934 |
glucose 1-dehydrogenase (NAD+) activity |
| Molecular Function |
GO:0047935 |
glucose 1-dehydrogenase (NADP+) activity |
| Molecular Function |
GO:0004345 |
glucose-6-phosphate dehydrogenase activity |
| Molecular Function |
GO:0050661 |
NADP binding |
| Biological Process |
GO:0006006 |
glucose metabolic process |
| Biological Process |
GO:0009051 |
pentose-phosphate shunt, oxidative branch |
| Biological Process |
GO:2000064 |
regulation of cortisol biosynthetic process |
| Biological Process |
GO:0097305 |
response to alcohol |
| Biological Process |
GO:0031667 |
response to nutrient levels |
Reference
[1] Yang Z, Yan C, Ma J, Peng P, Ren X et al.. Lactylome analysis suggests lactylation-dependent mechanisms of metabolic adaptation in hepatocellular carcinoma.. Nat Metab 5(1):61-79. 2023 Jan. PMID: 36593272.